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PWZ 029

  • PWZ-029
  • Chemical compound

    PWZ-029 is a benzodiazepine derivative drug with nootropic effects developed by WiSys, It acts as a subtype-selective, mixed agonist-inverse agonist at

    PWZ-029

    PWZ-029

    PWZ-029

  • Furosemide
  • Loop diuretic medication

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Furosemide

    Furosemide

    Furosemide

  • RDX
  • Explosive chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    RDX

    RDX

    RDX

  • Penicillin
  • Group of antibiotics derived from fungi

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Penicillin

    Penicillin

    Penicillin

  • Γ-Butyrolactone
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Γ-Butyrolactone

    Γ-Butyrolactone

    Γ-Butyrolactone

  • Baclofen
  • Gabapentinoid and Skeletal Muscle Relaxant

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Baclofen

    Baclofen

    Baclofen

  • Ciprofloxacin
  • Fluoroquinolone antibiotic

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Ciprofloxacin

    Ciprofloxacin

    Ciprofloxacin

  • 1,4-Butanediol
  • One of four stable isomers of butanediol

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    1,4-Butanediol

    1,4-Butanediol

    1,4-Butanediol

  • Lindane
  • Organochlorine chemical and an isomer of hexachlorocyclohexane

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Lindane

    Lindane

    Lindane

  • GABAA receptor negative allosteric modulator
  • Drug class

    Additional selective α5 subunit-containing GABAA receptor NAMs include PNV-001, PWZ-029, Ro4938581, and TB-21007. Certain drugs show weak GABAA receptor NAM activity

    GABAA receptor negative allosteric modulator

    GABAA_receptor_negative_allosteric_modulator

  • Xywav
  • Combination drug

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Xywav

    Xywav

  • Thujone
  • Group of four possible stereoisomers found in various plants: a.o., absinthe and mint

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Thujone

    Thujone

    Thujone

  • ASP-8062
  • Pharmaceutical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    ASP-8062

    ASP-8062

    ASP-8062

  • Glutamine
  • Amino acid

    kidney". Canadian Journal of Biochemistry. 57 (3): 233–237. doi:10.1139/o79-029. PMID 436006. DeBerardinis RJ, Mancuso A, Daikhin E, Nissim I, Yudkoff M

    Glutamine

    Glutamine

    Glutamine

  • Phenibut
  • CNS depressant medication

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Phenibut

    Phenibut

    Phenibut

  • Oenanthotoxin
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Oenanthotoxin

    Oenanthotoxin

    Oenanthotoxin

  • Piperidine-4-sulfonic acid
  • Pharmaceutical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Piperidine-4-sulfonic acid

    Piperidine-4-sulfonic acid

    Piperidine-4-sulfonic_acid

  • Clarithromycin
  • Antibiotic medication

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Clarithromycin

    Clarithromycin

    Clarithromycin

  • GABA
  • Main inhibitory neurotransmitter in the mammalian brain

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    GABA

    GABA

    GABA

  • Flumazenil
  • GABA receptor antagonist drug and benzodiazepine antidote

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Flumazenil

    Flumazenil

    Flumazenil

  • SH-053-R-CH3-2′F
  • Benzodiazepine drug

    also blocks the nootropic effects of the α5-selective inverse agonist PWZ-029, so amnesia is also a likely side effect. Replacement of the ester function

    SH-053-R-CH3-2′F

    SH-053-R-CH3-2′F

    SH-053-R-CH3-2′F

  • Pentylenetetrazol
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Pentylenetetrazol

    Pentylenetetrazol

    Pentylenetetrazol

  • Imipenem
  • Carbapenem antibiotic

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Imipenem

    Imipenem

    Imipenem

  • GABA receptor agonist
  • Category of drug

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    GABA receptor agonist

    GABA receptor agonist

    GABA_receptor_agonist

  • GABRA3
  • Protein-coding gene in humans

    dependence, and could make them superior to currently marketed drugs. Adipiplon PWZ-029 (partial agonist at α3, partial inverse agonist at α5) TP003 (Selective

    GABRA3

    GABRA3

    GABRA3

  • Levofloxacin
  • Antibiotic

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Levofloxacin

    Levofloxacin

    Levofloxacin

  • GABAA receptor
  • Ionotropic receptor and ligand-gated ion channel

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    GABAA receptor

    GABAA receptor

    GABAA_receptor

  • Tetramethylenedisulfotetramine
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Tetramethylenedisulfotetramine

    Tetramethylenedisulfotetramine

    Tetramethylenedisulfotetramine

  • Ofloxacin
  • Antibiotic to treat bacterial infections

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Ofloxacin

    Ofloxacin

    Ofloxacin

  • GABAergic
  • Affecting GABA systems in the brain

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    GABAergic

    GABAergic

  • Imidazoleacetic acid
  • Pharmaceutical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Imidazoleacetic acid

    Imidazoleacetic acid

    Imidazoleacetic_acid

  • Cicutoxin
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Cicutoxin

    Cicutoxin

    Cicutoxin

  • 4-AHP
  • Pharmaceutical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    4-AHP

    4-AHP

    4-AHP

  • N-Benzoyl-GABA
  • Pharmaceutical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    N-Benzoyl-GABA

    N-Benzoyl-GABA

    N-Benzoyl-GABA

  • Methylglyoxal
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Methylglyoxal

    Methylglyoxal

    Methylglyoxal

  • Γ-Hydroxybutyric acid
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Γ-Hydroxybutyric acid

    Γ-Hydroxybutyric acid

    Γ-Hydroxybutyric_acid

  • Picamilon
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Picamilon

    Picamilon

    Picamilon

  • Tutin (toxin)
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Tutin (toxin)

    Tutin (toxin)

    Tutin_(toxin)

  • GABRA2
  • Protein in humans

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    GABRA2

    GABRA2

    GABRA2

  • Thio-THIP
  • Pharmaceutical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Thio-THIP

    Thio-THIP

    Thio-THIP

  • Orenetide
  • Pharmaceutical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Orenetide

    Orenetide

    Orenetide

  • Dehydroepiandrosterone
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Dehydroepiandrosterone

    Dehydroepiandrosterone

    Dehydroepiandrosterone

  • IPTBO
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    IPTBO

    IPTBO

    IPTBO

  • BSPP (drug)
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    BSPP (drug)

    BSPP (drug)

    BSPP_(drug)

  • Picrotoxin
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Picrotoxin

    Picrotoxin

    Picrotoxin

  • JZP-386
  • Pharmaceutical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    JZP-386

    JZP-386

    JZP-386

  • Fipronil
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Fipronil

    Fipronil

    Fipronil

  • Oroxylin A
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Oroxylin A

    Oroxylin A

    Oroxylin_A

  • GABAA-rho receptor
  • Class of transport proteins

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    GABAA-rho receptor

    GABAA-rho_receptor

  • 2-Hydroxysaclofen
  • Chemical compound, GABA(B) receptor antagonist

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    2-Hydroxysaclofen

    2-Hydroxysaclofen

    2-Hydroxysaclofen

  • GABAA receptor agonist
  • Hallucinogenic drug

    (2004). "Gaboxadol". Drugs of the Future. 29 (5): 0449. doi:10.1358/dof.2004.029.05.803754. Retrieved 19 June 2025. Brickley SG, Mody I (January 2012). "Extrasynaptic

    GABAA receptor agonist

    GABAA receptor agonist

    GABAA_receptor_agonist

  • Γ-Valerolactone
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Γ-Valerolactone

    Γ-Valerolactone

    Γ-Valerolactone

  • Gabamide
  • Pharmaceutical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Gabamide

    Gabamide

    Gabamide

  • Ethyl acetoxy butanoate
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Ethyl acetoxy butanoate

    Ethyl acetoxy butanoate

    Ethyl_acetoxy_butanoate

  • Sodium oxybate
  • Medication to treat symptoms of narcolepsy

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Sodium oxybate

    Sodium oxybate

    Sodium_oxybate

  • 4-Fluorophenibut
  • GABAB receptor agonist and phenibut analogue

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    4-Fluorophenibut

    4-Fluorophenibut

    4-Fluorophenibut

  • Cyclothiazide
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Cyclothiazide

    Cyclothiazide

    Cyclothiazide

  • Flurothyl
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Flurothyl

    Flurothyl

    Flurothyl

  • Bemegride
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Bemegride

    Bemegride

    Bemegride

  • 11-Ketoprogesterone
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    11-Ketoprogesterone

    11-Ketoprogesterone

    11-Ketoprogesterone

  • FG-7142
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    FG-7142

    FG-7142

    FG-7142

  • Ionotropic GABA receptor
  • picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Ionotropic GABA receptor

    Ionotropic_GABA_receptor

  • Coriamyrtin
  • Convulsant toxin

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Coriamyrtin

    Coriamyrtin

    Coriamyrtin

  • Thiomuscimol
  • Pharmaceutical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Thiomuscimol

    Thiomuscimol

    Thiomuscimol

  • Α5IA
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Α5IA

    Α5IA

    Α5IA

  • 4-PIOL
  • Pharmaceutical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    4-PIOL

    4-PIOL

    4-PIOL

  • Homotaurine
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Homotaurine

    Homotaurine

    Homotaurine

  • Loreclezole
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Loreclezole

    Loreclezole

    Loreclezole

  • EBOB
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    EBOB

    EBOB

    EBOB

  • Valiloxybate
  • Pharmaceutical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Valiloxybate

    Valiloxybate

    Valiloxybate

  • 4-Amino-1-butanol
  • Organic compound and GABA analogue and precursor

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    4-Amino-1-butanol

    4-Amino-1-butanol

  • N-Acetyl-γ-aminobutyric acid
  • Endogenous GABA precursor

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    N-Acetyl-γ-aminobutyric acid

    N-Acetyl-γ-aminobutyric acid

    N-Acetyl-γ-aminobutyric_acid

  • Cetyl-GABA
  • Pharmaceutical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Cetyl-GABA

    Cetyl-GABA

  • Isoguvacine
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Isoguvacine

    Isoguvacine

    Isoguvacine

  • Aceburic acid
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Aceburic acid

    Aceburic acid

    Aceburic_acid

  • Monastrol
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Monastrol

    Monastrol

    Monastrol

  • Tolgabide
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Tolgabide

    Tolgabide

    Tolgabide

  • Ro15-4513
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Ro15-4513

    Ro15-4513

    Ro15-4513

  • L-655,708
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    L-655,708

    L-655,708

    L-655,708

  • Pregnanolone
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Pregnanolone

    Pregnanolone

    Pregnanolone

  • Gabazine
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Gabazine

    Gabazine

    Gabazine

  • GABRA5
  • Protein found in humans

    trials for treating cognitive deficit in Down syndrome. L-655,708 MRK-016 PWZ-029: moderate inverse agonist Pyridazines Ro4938581 TB-21007 GABAA receptor

    GABRA5

    GABRA5

    GABRA5

  • Ibotenic acid
  • Naturally occurring glutamate receptor agonist neurotoxin

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Ibotenic acid

    Ibotenic acid

    Ibotenic_acid

  • Bupleurotoxin
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Bupleurotoxin

    Bupleurotoxin

  • Hopantenic acid
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Hopantenic acid

    Hopantenic acid

    Hopantenic_acid

  • Hydrastine
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Hydrastine

    Hydrastine

    Hydrastine

  • List of benzodiazepines
  • 5-a]pyrrolo[2,1-c] [1,4]benzodiazepine-1-carboxylate 5311203 130477-52-0 PWZ-029 8-chloro-3-(methoxymethyl)-5-methyl-4H-imidazo[1,5-a] [1,4]benzodiazepin-6-one

    List of benzodiazepines

    List of benzodiazepines

    List_of_benzodiazepines

  • SL-75102
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    SL-75102

    SL-75102

    SL-75102

  • Gaboxadol
  • Chemical compound

    (2004). "Gaboxadol". Drugs of the Future. 29 (5): 0449. doi:10.1358/dof.2004.029.05.803754. Retrieved 19 June 2025. "Gaboxadol - Lundbeck A/S". AdisInsight

    Gaboxadol

    Gaboxadol

    Gaboxadol

  • ADX-71441
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    ADX-71441

    ADX-71441

    ADX-71441

  • Prasterone
  • Medical usage of the prasterone compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Prasterone

    Prasterone

    Prasterone

  • Nefiracetam
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Nefiracetam

    Nefiracetam

    Nefiracetam

  • 5β-Dihydroprogesterone
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    5β-Dihydroprogesterone

    5β-Dihydroprogesterone

    5β-Dihydroprogesterone

  • N-Acetylputrescine
  • Endogenous GABA precursor

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    N-Acetylputrescine

    N-Acetylputrescine

    N-Acetylputrescine

  • Levomethorphan
  • Opioid analgesic

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Levomethorphan

    Levomethorphan

    Levomethorphan

  • Ro 19-4603
  • Benzodiazepine antagonist

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Ro 19-4603

    Ro 19-4603

    Ro_19-4603

  • PNV-001
  • Pharmaceutical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    PNV-001

    PNV-001

  • GABA receptor antagonist
  • Drug Class

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    GABA receptor antagonist

    GABA_receptor_antagonist

  • Isopregnanolone
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Isopregnanolone

    Isopregnanolone

    Isopregnanolone

  • Sarmazenil
  • Chemical compound

    picrotoxinin and dihydropicrotoxinin) PNV-001 Pregnenolone sulfate Propybicyphat PWZ-029 Radequinil Ro 15-4513 Ro 19-4603 RO4882224 RO4938581 Sarmazenil SCS Suritozole

    Sarmazenil

    Sarmazenil

    Sarmazenil

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  • Paz
  • Boy/Male

    Hebrew, Hindu, Indian, Marathi, Parsi, Spanish

    Paz

    Peace

    Paz

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Online names & meanings

  • Maaniky
  • Boy/Male

    Hindu, Indian

    Maaniky

    Yeda

  • Kumarika | குமாரிகா
  • Girl/Female

    Tamil

    Kumarika | குமாரிகா

    Young girl, Jasmine

  • BRANISLAV
  • Male

    Czechoslovakian

    BRANISLAV

    , glorious protector.

  • Arul
  • Boy/Male

    Assamese, Hindu, Indian, Kannada, Marathi, Tamil, Telugu

    Arul

    God's Grace; Gods Blessing

  • Hafeezah
  • Girl/Female

    Muslim/Islamic

    Hafeezah

    Keeper of the sacred book

  • POMPEO
  • Male

    Italian

    POMPEO

    Italian form of Roman Latin Pompeius, possibly POMPEO means "display, solemn procession." 

  • Mustin
  • Surname or Lastname

    English (West Midlands)

    Mustin

    English (West Midlands) : origin uncertain; possibly a variant of Muston or perhaps of Musto.

  • Naajy | ناجی
  • Boy/Male

    Muslim

    Naajy | ناجی

    Safe

  • Vimalbir
  • Boy/Male

    Indian, Punjabi, Sikh

    Vimalbir

    Pure and Brave

  • Sashriti
  • Boy/Male

    Hindu, Indian, Malayalam, Marathi

    Sashriti

    Protector of Wealth

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PWZ 029

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